DOI: 10.1039/d3md00044c ISSN: 2632-8682

Enhancing allosteric inhibition of dihydrodipicolinate synthase through the design and synthesis of novel dimeric compounds

Rebecca M. Christoff, Mohammad Al Bayer, Tatiana P. Soares da Costa, Matthew A. Perugini, Belinda M. Abbott
  • Organic Chemistry
  • Drug Discovery
  • Pharmaceutical Science
  • Pharmacology
  • Molecular Medicine
  • Biochemistry

The synthesis of the first low micromolar dimeric inhibitor of E. coli DHDPS is reported.

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