DOI: 10.1039/d3ob01147j ISSN: 1477-0520

Aryne and CO2-based formal [2 + 2 + 2] annulation to access tetrahydroisoquinoline-fused benzoxazinones

Shiqi Liu, Kun Zhang, Yutong Meng, Jiaxi Xu, Ning Chen
  • Organic Chemistry
  • Physical and Theoretical Chemistry
  • Biochemistry

A three-component formal [2 + 2 + 2] annulation has been described from 3,4-dihydroisoquinolines, CO2, and benzynes, accessing tetrahydroisoquinoline-fused benzoxazinones in moderate to excellent yields.

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