DOI: 10.1039/d3md00286a ISSN: 2632-8682

α-Aminophosphonate inhibitors of metallo-β-lactamases NDM-1 and VIM-2

Katarzyna Palica, Fritz Deufel, Susann Skagseth, Gabriela Paula Di Santo Metzler, Johannes Thoma, Anna Andersson Rasmussen, Arto Valkonen, Per Sunnerhagen, Hanna-Kirsti S. Leiros, Hanna Andersson, Mate Erdelyi
  • Organic Chemistry
  • Drug Discovery
  • Pharmaceutical Science
  • Pharmacology
  • Molecular Medicine
  • Biochemistry

α-Aminophosphonate inhibitors of the bacterial metallo-β-lactamases NDM-1 and VIM-2 have been developed and studied.

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