DOI: 10.1039/d6ra06655k ISSN: 2046-2069

Targeting DYRK1A with rationally designed pyrazine–guanidine hybrids for Alzheimer's disease: design, synthesis, and biological evaluation

Sabiha Khan, Sumaiya Khan, Shafa Khan, Md. Ataur Rahman, Abdur Rahman, Aquib Reza, Shilpi Khurana, Mohammad Zahid Ashraf, Asimul Islam, Nasimul Hoda

Novel pyrazine–guanidine hybrids as potent DYRK1A inhibitors for Alzheimer's disease.