DOI: 10.1039/d6ra03053j ISSN: 2046-2069
Hybrid amine-derived compounds as cytotoxic anticancer leads: design, synthesis, and biological evaluation
Reem Odeh, Areej M. Jaber, Mazen Al-Sulaibi, Hamdi Nsairat, Mutasem O. TahaNovel amine-based hybrid compounds were synthesized and evaluated as Aurora-A kinase inhibitors. Compound 8a showed the strongest activity and significant cytotoxicity against A549 lung cancer cells, highlighting its potential as an anticancer lead.