DOI: 10.1039/d3ob00985h ISSN:

Electrochemical bromocyclization enables 3,5-diversification of heterocyclic indolines

Hai Ren, Rui-An Wang, Jun Shi, Jun-Rong Song, Wei Wu, Qin Chi, Ni Zhang
  • Organic Chemistry
  • Physical and Theoretical Chemistry
  • Biochemistry

We report a protonic-acid-promoted electrosynthetic strategy for the dearomative dibromocyclization of tryptamine/tryptophol derivatives for the convenient late-stage 3,5-diversification of heterocyclic indolines.

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