DOI: 10.1039/d3ob01934a ISSN: 1477-0520

Copper-catalyzed oxidative cyclization of 2-(1H-pyrrol-1-yl)aniline and alkylsilyl peroxides: a route to pyrrolo[1,2-a]quinoxalines

Zhenyu An, Man Miao, Fengkai Sun, Xiao-Bing Lan, Jian-Qiang Yu, Xiaoli Guo, Jian Zhang
  • Organic Chemistry
  • Physical and Theoretical Chemistry
  • Biochemistry

An efficient method was developed for the one-pot construction of pyrrolo[1,2-a]quinoxalines via a Cu(

ii
)-catalyzed domino reaction between 2-(1H-pyrrol-1-yl)anilines and alkylsilyl peroxides.

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