DOI: 10.1039/d6cc04631b ISSN: 1359-7345
Copper-catalyzed C(sp 3 )–H amination for direct N -alkylation of β-enamines using ethers and alkanes
Chengli Deng, Jiarui Wu, Zijing Bai, Fan Yang, Yefeng Zhu, Peng Gao, Wei ShiSelective N -alkylation of β-enamines with ethers and alkanes has been investigated via a copper-catalyzed C(sp 3 )–H amination transformation.