DOI: 10.4103/ijp.ijp_1281_25 ISSN: 0253-7613

Combinatorial effects of curcumin, morin, and phyllanthin in MDA-MB-231 and MCF-7 breast cancer cell lines

Sowmya Vuppaladadium, Joseph Xavier, Alanka Ketan Kumar, Sandhya Annamaneni

Abstract:

OBJECTIVES:

To evaluate the cytotoxic efficacy and interaction dynamics of curcumin, morin, and phyllanthin – individually and in dual (C + M) and triple (C + M + P) combinations – in estrogen receptor-positive (MCF-7) and triple-negative (MDA-MB-231) breast cancer cell lines.

MATERIALS AND METHODS:

Cytotoxicity was assessed by MTT assay after 24 h of treatment with varying concentrations of the phytochemicals. Half-maximal inhibitory concentrations were determined, and interaction effects were analyzed using the Combination Index (CI) model. Two-way ANOVA was used to quantify compound contributions and the statistical significance of interactions.

RESULTS:

The Curcumin + Morin (C + M) combination exhibited additive cytotoxic effects in both MDA-MB-231 (CI = 0.881) and MCF-7 (CI = 0.860) cells, showing significant dose-dependent inhibition ( P < 0.001). Addition of phyllanthin (C + M + P) further enhanced cytotoxicity, resulting in additive interaction in MDA-MB-231 (CI = 0.864) and synergistic interaction in MCF-7 (CI = 0.684). Contribution analysis indicated that phyllanthin, despite low individual potency, accounted for approximately 50%–55% of total cytotoxicity by amplifying the effects of curcumin and morin.

CONCLUSIONS:

Combinations of curcumin, morin, and phyllanthin demonstrate subtype-dependent cytotoxic enhancement, with synergy evident in hormone receptor-positive breast cancer cells. These findings support the potential of phytochemical co-treatment as a complementary approach to improve therapeutic efficacy through multi-pathway modulation while minimizing toxicity.

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