DOI: 10.1039/d6sc03753d ISSN: 2041-6520
Chemically triggered bioorthogonal activation of antimicrobial peptide mimic prodrugs
Hao Luo, Rhiannon P. Kuchel, Kevin Neumann, Edgar H. H. WongA new antimicrobial peptide-mimicking prodrug is developed here, which can be activated precisely by a chemical trigger via click chemistry to combat multidrug-resistant bacteria effectively.