DOI: 10.3390/ijms27135947 ISSN: 1422-0067

A Multi-Engine Consensus Docking Pipeline for RNA Aptamer Screening Against ACC Oxidase (ACO): Statistical Validation, Machine Learning Analysis, and Pilot Cross-Target Evaluation Against ACC Synthase (ACS)

Héctor Ramón Martínez-de la Hoya, Cristian Patricia Cabrales-Arellano, Josué Ortiz-Medina, Efren Delgado, Juan Antonio Rojas-Contreras, Norma A. García-Vidaña, Damián Reyes-Jáquez, Rubén Guerrero-Rivera

Postharvest losses in climacteric fruits are largely driven by ethylene, and inhibiting its biosynthesis is an active research goal. RNA aptamers are attractive candidates for modulating the two rate-limiting enzymes—ACC oxidase (ACO) and ACC synthase (ACS), without the toxicity concerns of chemical inhibitors. We built a computational pipeline using three independent docking engines: ITD DOCK (Graphics Processing Unit [GPU]-accelerated, Assisted Model Building with Energy Refinement [AMBER] force fields), HDOCK Lite (knowledge-based geometric potentials), and HADDOCK3 (semi-flexible refinement), screened against large aptamer libraries. Applied to ACC oxidase with 9813 aptamers, engine scores were largely complementary, with all pairwise correlations statistically non-significant on the full dataset (Spearman |ρ|≤0.013, p>0.20 for all pairs, n=9813). A Random Forest on sequence-only features failed to predict docking scores (R2=−0.012, Root Mean Square Error [RMSE] = 21.79 kcal/mol), while a positive-control model on HADDOCK3 energy components achieved R2=0.991, confirming that predictive information only becomes available after docking. A preliminary pilot screening against ACC synthase (n=97 valid complexes) suggested pipeline generalizability to a second structurally distinct target and identified two putative dual-active candidates, pending confirmation against the full library. The complete workflow is automated in AptaDock, a standalone desktop application.

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