DOI: 10.1002/jhet.4932 ISSN: 0022-152X
Synthesis of 5‐Aryltetrahydrobenzazepines
Naveenkumar Thoti, Deepika Gupta, Heera Lal, Indrapal Singh AidhenABSTRACT
Envisaging 5‐aryltetrahydrobenzazepinone and 5‐aryltetrahydrobenzazepines as conformationally locked potential B0AT1 inhibitors, a convenient synthetic route has been developed for their access. The synthetic route banks on using the Schmidt reaction for quick access to symmetrical/unsymmetrical 5‐aryltetrahydrobenzazepinone and 5‐aryltetrahydrobenzazepines.